Irisin (FNDC5 hormone form)

Class Peptide hormone (myokine)Receptor Integrin-associated receptor signaling

Function

Irisin is a peptide signaling hormone involved in energy metabolism, skeletal muscle communication, thermogenic adaptation, mitochondrial regulation, and metabolic signaling between muscle and adipose tissue. The hormone is released during muscular activity and participates in communication pathways linking physical movement with systemic metabolic adaptation.

Irisin influences energy expenditure, mitochondrial biogenesis, glucose utilization, lipid metabolism, and thermogenic gene expression within adipose tissue. The hormone also contributes to skeletal muscle signaling, bone communication pathways, and regulation of metabolic flexibility during changing energy demands. Through these actions, irisin functions as an endocrine messenger connecting muscular activity with whole-body metabolic physiology.

Production

Irisin is produced mainly by skeletal muscle through cleavage of the membrane protein FNDC5. Production increases during muscular contraction and exercise-associated signaling. Additional expression occurs in adipose tissue, heart tissue, nervous system structures, and additional metabolic organs.

The hormone is released into circulation where it can act on adipose tissue, skeletal muscle, bone, and additional endocrine-responsive tissues. Local muscle production therefore serves as a key interface between physical activity and endocrine metabolic communication.

Regulation

Irisin production is regulated by muscular activity, PGC-1alpha signaling, mitochondrial demand, energy metabolism, exercise physiology, oxidative stress pathways, and nutrient availability. Endurance-associated signaling strongly influences FNDC5 expression and irisin release.

Irisin acts through signaling systems associated with thermogenic gene expression, mitochondrial adaptation, metabolic regulation, and adipocyte communication pathways. Interactions with AMPK signaling, oxidative metabolism pathways, and mitochondrial biogenesis systems contribute to its physiological effects. Through these integrated muscle-endocrine signaling systems, irisin coordinates metabolic adaptation, energy expenditure, mitochondrial regulation, and communication between skeletal muscle and peripheral metabolic tissues.

Identity & Secretion

Primary Source GlandSkeletal muscle
Secretion PatternExercise-inducible secretion pattern
PrecursorFNDC5 precursor protein

Nutrient Requirements

Nutrient Precursors
  • Amino acids from dietary protein required for synthesis
Required Vitamins
  • B vitamins; vitamin C (general metabolic and collagen milieu)
Required Minerals
  • Magnesium; potassium (general metabolic roles)

Key Foods

  • Legumes; soy foods; quinoa; oats; leafy greens; berries; nuts; seeds

Targets & Signaling

Target Tissues
  • Adipose tissue; muscle; bone; liver; nervous system (reported in research)
Feedback Loops
  • Exercise training upregulates PGC-1alpha -> FNDC5 -> irisin
Second Messengers
  • Integrin-linked kinase signaling cascades
Pathways Involved
  • MAPK/ERK and p38 pathways linked to integrin signaling

Key Functions

  • Supports metabolic flexibility and energy expenditure signaling

Plant-Based Focus

  • Whole-food plant-based diet supports metabolic efficiency and muscle recovery

Clinical Context

Assay Notes
Assay variability reported in irisin quantification research

Linked Knowledge

Phytochemicals
  • Quercetin; catechins; resveratrol (exercise-adaptive phytochemical contexts)
Amino Acids
  • Leucine; arginine (amino acids relevant to muscle metabolism)
Foods
  • Soy foods; legumes; quinoa; oats; leafy greens; berries; nuts; seeds
Vitamins
  • B-complex; vitamin C
Minerals
  • Magnesium; potassium
Ailments
  • Sedentary lifestyle context (non-medical informational)

Dietary Modulators

  • Regular physical activity and muscle use support beneficial expression

Inhibitors / Activators

Inhibitors
  • Physical inactivity can reduce endogenous adaptive signaling (context only)

Summary

Exercise-stimulated myokine involved in metabolic adaptation signaling

SUMMARY OF EFFECTS ON THE BODY

Helps coordinate the beneficial systemic effects of movement and diet patterns

Research

Research reviews discussing PGC1-alpha to FNDC5 cleavage and integrin signaling
Created: Nov 11, 2025 Updated: May 27, 2026